SCHEMBL7969712

SCHEMBL7969712

O=c1[nH]c2ccc(-n3ccnc3)cc2n2cncc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.47
PDE3B Q13370 3/20 0.44
PDE3A Q14432 3/20 0.44
CRBN Q96SW2 2/20 0.44
TBXAS1 P24557 1/20 0.44
IDH1 O75874 1/20 0.43
CYP19A1 P11511 2/20 0.42
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
CHEK1 O14757 1/20 0.41
IDO1 P14902 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PDE2A O00408 2/20 0.40
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39
GRIK1 P39086 1/20 0.39
GRIA1 P42261 1/20 0.39
GRIA2 P42262 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7268865 0.81 GRIA1 (0.53) PGRPDE3BPDE3ACRBNTBXAS1
SCHEMBL7269285 0.78 PGR (0.44) PGRPDE3BPDE3ACRBNTBXAS1
SCHEMBL8911996 0.78 PGR (0.51) PGRPDE3BPDE3ACRBNTBXAS1
SCHEMBL21676341 0.78 GRIK1 (0.52) PGRPDE3BPDE3ACRBNTBXAS1
Hydrochloric Acid SCHEMBL8130929 0.77 PGR (0.47) PGRPDE3BPDE3ACRBNTBXAS1
SCHEMBL7268386 0.76 PDE4A (0.51) PGRPDE3BPDE3ACRBNTBXAS1
SCHEMBL2468642 0.75 DAO (0.46)
SCHEMBL7982949 0.75 GABRA5 (0.36) CHEK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL29235466 0.75 TP53 (0.46) CHEK1IDO1
SCHEMBL7980241 0.75 DAO (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed