SCHEMBL7971124

SCHEMBL7971124

COC(=O)c1ccc2cnn(C3CCCC3)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
NPSR1 Q6W5P4 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ATM Q13315 1/20 0.50
HTR1A P08908 1/20 0.48
HTR1B P28222 1/20 0.48
HTR1F P30939 1/20 0.48
KDM4E B2RXH2 4/20 0.48
HPGD P15428 2/20 0.48
LMNA P02545 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
RPS6KB1 P23443 1/20 0.43
MERTK Q12866 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
POLB P06746 1/20 0.42
APOBEC3A P31941 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30040346 0.95 HTR1A (0.50) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A
SCHEMBL23467071 0.90 ALDH1A1 (0.50) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A
SCHEMBL24338759 0.89 HTR1A (0.46) ALDH1A1HTR1AHTR1BHTR1FHPGD
SCHEMBL31403635 0.87 RPS6KB1 (0.48) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A
SCHEMBL24339264 0.86 HTR1A (0.43) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A
SCHEMBL30174436 0.86 HTR1A (0.43) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A
SCHEMBL7419168 0.85 HCAR3 (0.56) ALDH1A1HTR1AHTR1BHTR1FHPGD
SCHEMBL24900263 0.84 RXRA (0.50) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A
SCHEMBL3605908 0.84 HTR1A (0.44) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A
SCHEMBL904780 0.84 CYP11B1 (0.47) ALDH1A1NPSR1SMN1; SMN2ATMHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6262040-B1 Indazole derivatives and their use as inhibitors of phosphodiesterase (PDE) type IV and the production of tumor necrosis factor (TNF) PFIZER INC 2001-07-17 US disclosed
CN-1234031-A Indazole derivatives and their use as inhibitors of phosphodiesterase (PDE) type IV and the prodn. of tumor necrosis factor (TNF) PFIZER (US) 1999-11-03 CN disclosed