SCHEMBL7973080

SCHEMBL7973080

COc1c2c(c(OC)c(OC)c1OC)CC(CCCCCCCCN1CCC(N3CCCCC3)CC1)C2

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.42
HRH3 Q9Y5N1 7/20 0.42
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
ABCB1 P08183 1/20 0.37
CHRM5 P08912 1/20 0.37
ADRA2A P08913 1/20 0.37
CHRM1 P11229 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
CHRM3 P20309 1/20 0.37
KCNH2 Q12809 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
AVPR2 P30518 1/20 0.37
AVPR1A P37288 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7971226 0.81 HRH3 (0.42) SIGMAR1HRH3CHRM2CHRM1
SCHEMBL7977198 0.78 ALDH1A1 (0.43) SIGMAR1HRH3CHRM2CHRM1KCNH2
SCHEMBL7961213 0.77 HRH3 (0.57) HRH3
Hydrochloric Acid SCHEMBL7971441 0.77 HRH3 (0.56) HRH3
Hydrochloric Acid SCHEMBL7977428 0.75 SIGMAR1 (0.52) SIGMAR1CYP3A4
Hydrochloric Acid SCHEMBL7974723 0.71 CCR3 (0.49) SIGMAR1
SCHEMBL19494839 0.71 GNAO1 (0.56) HRH3KCNH2
SCHEMBL7974667 0.71 L3MBTL3 (0.53)
SCHEMBL24218139 0.69 GNAO1 (0.53) HRH3
SCHEMBL10025501 0.68 HRH3 (0.55) HRH3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326369-B1 ALZHEIMER'S DISEASE TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 2001-12-04 US disclosed