SCHEMBL7974338

SCHEMBL7974338

CCCCc1ccccc1S(=O)(=O)Nc1ncnc(Cl)c1-c1ccc(C)cc1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 2/20 0.41
PKM P14618 1/20 0.38
ALDH1A1 P00352 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CCR4 P51679 1/20 0.37
EDNRB P24530 2/20 0.37
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9044020 0.96 EDNRA (0.42) EDNRAPKMALDH1A1RXFP1L3MBTL1
SCHEMBL9491423 0.91 EDNRA (0.43) EDNRAPKMALDH1A1RXFP1L3MBTL1
SCHEMBL9047803 0.83 PKM (0.55) EDNRAPKMALDH1A1RXFP1L3MBTL1
SCHEMBL9045446 0.82 KIT (0.48) EDNRAALDH1A1EDNRBMEN1MAPT
SCHEMBL9043342 0.79 EDNRA (0.64) EDNRAEDNRB
SCHEMBL9044797 0.79 RXFP1 (0.54) RXFP1
SCHEMBL9043805 0.78 EDNRA (0.49) EDNRAALDH1A1EDNRBMEN1MAPT
SCHEMBL9045052 0.77 MEN1 (0.55) EDNRAALDH1A1EDNRBMEN1MAPT
SCHEMBL14289222 0.77 EDNRA (0.42) EDNRAALDH1A1EDNRBMEN1MAPT
SCHEMBL9043154 0.77 ALDH1A1 (0.44) EDNRAPKMALDH1A1RXFP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001081335-A1 PYRIMIDINE-SULFONAMIDES HAVING ENDOTHELIN-ANTAGONIST ACTIVITY ACTELION PHARMACEUTICALS LTD (CH) 2001-11-01 WO disclosed