SCHEMBL7975606

SCHEMBL7975606

Cc1ccc(-c2n[nH]c(-c3nc4cc5c(cc4[nH]3)CNC5)c2OC(=O)N2CCCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.37
ATR Q13535 4/20 0.35
HCRTR1 O43613 4/20 0.35
HCRTR2 O43614 4/20 0.35
CHEK2 O96017 3/20 0.34
ACHE P22303 2/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CNR1 P21554 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7960176 0.99 BRD4 (0.36) BRD4ATRHCRTR1HCRTR2CHEK2
SCHEMBL7960886 0.85 CNR1 (0.38) BRD4ATRCHEK2ACHESIRT2
SCHEMBL7972878 0.85 HPSE (0.38) BRD4CHEK2RAB9ASMN1; SMN2NPC1
SCHEMBL10140034 0.84 CNR1 (0.39) BRD4ATRCHEK2ACHESIRT2
SCHEMBL7975112 0.78 F9 (0.47) BRD4CHEK2RAB9ASMN1; SMN2CNR1
SCHEMBL10140037 0.78 CYP2C9 (0.41) BRD4ATRACHESIRT2SIRT1
SCHEMBL20307729 0.74 F9 (0.40) CHEK2RAB9ASMN1; SMN2NPC1
SCHEMBL7969308 0.74 TSPO (0.37) BRD4CHEK2SIRT2SIRT1
SCHEMBL7980011 0.73 CHEK2 (0.38) BRD4ATRCHEK2RAB9ASMN1; SMN2
SCHEMBL7960749 0.73 HDAC3 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed