SCHEMBL7975959

SCHEMBL7975959

CCN(CC)C(=O)Cc1c(-c2ccc(CN3CCOCC3)cc2)n[nH]c1-c1nc2cc(C(=N)N)ccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 7/20 0.45
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
CDK7 P50613 3/20 0.42
PARP1 P09874 1/20 0.40
AURKA O14965 5/20 0.39
AURKB Q96GD4 5/20 0.39
CDK1 P06493 4/20 0.39
CCNB1 P14635 4/20 0.39
CDK2 P24941 4/20 0.39
SLC2A1 P11166 1/20 0.39
F9 P00740 1/20 0.38
F10 P00742 1/20 0.38
F11 P03951 1/20 0.38
F7 P08709 1/20 0.38
FGFR1 P11362 2/20 0.37
FGFR2 P21802 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10140130 0.78 HDAC3 (0.43) CHEK1HDAC3HDAC1HDAC2HDAC8
SCHEMBL16258968 0.76 HDAC3 (0.42) CHEK1HDAC3HDAC1HDAC2HDAC8
SCHEMBL7974939 0.73 HDAC6 (0.59) CHEK1HDAC3HDAC1HDAC2HDAC8
SCHEMBL7960749 0.71 HDAC3 (0.43) CHEK1HDAC3HDAC1HDAC2HDAC8
SCHEMBL7973134 0.70 F10 (0.64) HDAC3HDAC1HDAC8HDAC6F9
SCHEMBL10139999 0.70 HDAC6 (0.54) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL7969308 0.70 TSPO (0.37) KDRSYK
SCHEMBL18229740 0.69 HDAC6 (0.84) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL7960699 0.68 F10 (0.67) F9F10F11F7MAPKAPK5
SCHEMBL20307774 0.68 F10 (0.67) F9F10F11F7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed