SCHEMBL7976189

SCHEMBL7976189

COc1ccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4cccc(Cl)c34)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 3/20 0.40
CDK7 P50613 3/20 0.40
CDK9 P50750 3/20 0.40
CCNH P51946 3/20 0.40
MNAT1 P51948 3/20 0.40
CCNE1 P24864 2/20 0.40
CDK2 P24941 2/20 0.40
MAOB P27338 1/20 0.36
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNB3 Q05901 1/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
CYP2D6 P10635 1/20 0.35
KCNH2 Q12809 1/20 0.35
HTR6 P50406 1/20 0.35
TGFBR1 P36897 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990422 0.93 ABL1 (0.38) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7990432 0.91 CDK9 (0.42) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7990707 0.91 CDK9 (0.44) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7976643 0.87 CDK9 (0.40) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7511168 0.86 CHEK1 (0.40) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7986667 0.86 CDK7 (0.44) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7993811 0.85 KDR (0.39) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7991016 0.84 CCNT1 (0.37) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7976151 0.84 CCNT1 (0.37) CCNT1CDK7CDK9CCNHMNAT1
SCHEMBL7987194 0.84 HTR6 (0.37) CCNT1CDK7CDK9CCNHMNAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed