SCHEMBL7990422

SCHEMBL7990422

COc1cccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4cccc(Cl)c34)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.38
EGFR P00533 3/20 0.38
SRC P12931 3/20 0.38
ABL2 P42684 3/20 0.38
CCNT1 O60563 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
CCNH P51946 1/20 0.38
MNAT1 P51948 1/20 0.38
CYP2C19 P33261 1/20 0.36
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
CYP2D6 P10635 1/20 0.35
KCNH2 Q12809 1/20 0.35
EED O75530 1/20 0.35
CHEK1 O14757 2/20 0.34
CYP11B1 P15538 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976189 0.93 CCNT1 (0.40) EGFRSRCCCNT1CCNE1CDK2
SCHEMBL7976643 0.90 CDK9 (0.40) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7990707 0.90 CDK9 (0.44) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7976272 0.87 CCNT1 (0.41) ABL1EGFRSRCABL2CCNT1
SCHEMBL7990432 0.87 CDK9 (0.42) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7986731 0.87 CHEK1 (0.41) ABL1EGFRSRCABL2CYP2C19
SCHEMBL7994923 0.86 PRKCA (0.40) ABL1EGFRSRCABL2CCNT1
SCHEMBL7990984 0.86 CCNT1 (0.36) ABL1EGFRSRCABL2CCNT1
SCHEMBL7975970 0.86 HTR6 (0.39) ABL1EGFRSRCABL2CYP2C19
SCHEMBL7993811 0.84 KDR (0.39) CCNT1CCNE1CDK2CDK7CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed