SCHEMBL7273301

SCHEMBL7273301

CNCCCCCCN1CNc2ccncc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC22A2 O15244 1/20 0.32
SLC22A1 O15245 1/20 0.32
SLC22A3 O75751 1/20 0.32
CYP1A2 P05177 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
DRD2 P14416 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
NFKB1 P19838 1/20 0.32
CHRM3 P20309 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
MAPK1 P28482 1/20 0.32
SLC6A4 P31645 1/20 0.32
ADRA1A P35348 1/20 0.32
HRH1 P35367 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14185922 0.76 SLC6A2 (0.53) CYP3A4CYP2D6SLC6A2SLC22A2SLC22A1
SCHEMBL7977462 0.69 GAA (0.35) CYP3A4CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL9038711 0.65 CES1 (0.44) CYP2D6CYP1A2HTTMEN1KMT2A
SCHEMBL7267151 0.63 DAO (0.47) MAPK1HTTSMN1; SMN2
SCHEMBL24669482 0.62 USP2 (0.32) CYP3A4CYP2D6HTT
SCHEMBL24719048 0.61 MEN1 (0.42) CYP3A4CYP2D6SLC6A2SLC22A2SLC22A1
SCHEMBL8091908 0.61 BRPF1 (0.41) CYP2D6CYP1A2CHRM2CHRM1DRD2
SCHEMBL6283776 0.61 KMT2A (0.43) CYP3A4CYP2D6CYP1A2MEN1KMT2A
SCHEMBL7975285 0.61 PDE9A (0.32) CACNA1BCHRNB2CHRNA4
SCHEMBL10541053 0.60 POLB (0.46) HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268148-B1 TETRAHYDRONAPHTHALENE DERIVATIVES AND MEDICAMENTS CONTAINING THEM F. HOFFMANN-LA ROCHE AG (CH) 1991-12-11 EP disclosed