SCHEMBL7978560

SCHEMBL7978560

COC(=O)Nc1nc(N)nc(-c2ccccc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.52
ADORA3 P0DMS8 2/20 0.51
ADORA2A P29274 2/20 0.51
ADORA2B P29275 2/20 0.51
ADORA1 P30542 2/20 0.51
POLB P06746 1/20 0.51
TPH1 P17752 6/20 0.47
TSHR P16473 3/20 0.47
USP2 O75604 1/20 0.47
ALDH1A1 P00352 2/20 0.46
ALOX15 P16050 2/20 0.46
LMNA P02545 2/20 0.46
GAA P10253 1/20 0.46
MAPK1 P28482 1/20 0.46
HSP90AA1 P07900 1/20 0.45
HSP90AB1 P08238 1/20 0.45
KDM4E B2RXH2 1/20 0.45
PKM P14618 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7244671 0.89 ALDH1A1 (0.51) NPSR1ADORA3ADORA2AADORA1TSHR
SCHEMBL2229906 0.83 NPSR1 (0.56) NPSR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL6982880 0.82 TPH1 (0.56) NPSR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7981524 0.82 RAB9A (0.47) NPSR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL3945635 0.82 ADORA1 (0.60) NPSR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7978506 0.81 ALDH1A1 (0.46) NPSR1ADORA3ADORA1TPH1TSHR
Benzoguanamine SCHEMBL8849771 0.80 ADORA1 (0.61) NPSR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL7776751 0.79 LMNA (0.40) NPSR1TSHRALDH1A1ALOX15LMNA
SCHEMBL5159281 0.78 NPSR1 (0.54) NPSR1ADORA3ADORA2AADORA2BADORA1
SCHEMBL3133857 0.77 TPH1 (0.60) NPSR1ADORA3ADORA1TPH1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6197957-B1 CATALYTIC REACTION WITH CARBON MONOXIDE CYTEC TECHNOLOGY CORP. 2001-03-06 US disclosed
EP-0649842-B1 Process for preparing derivatives of (halo)amino compounds by carbonylation CYTEC TECH CORP (US) 1998-06-03 EP disclosed
EP-0649842-A1 Process for preparing derivatives of (halo)amino compounds by carbonylation CYTEC TECHNOLOGY CORP. (US) 1995-04-26 EP disclosed