SCHEMBL7978561

SCHEMBL7978561

COC(=O)[C@@H]1Cc2ccccc2CN1C(=O)C(=O)c1cccs1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 3/20 0.43
MMP1 P03956 2/20 0.43
ADAM17 P78536 2/20 0.43
MMP3 P08254 1/20 0.43
ADAM9 Q13443 1/20 0.43
NR1D1 P20393 3/20 0.42
F10 P00742 1/20 0.42
POLB P06746 1/20 0.40
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CASP1 P29466 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
PTPN1 P18031 1/20 0.39
SLC18A3 Q16572 1/20 0.38
HSD17B10 Q99714 2/20 0.38
NPC1 O15118 1/20 0.38
USP2 O75604 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978564 1.00 MMP9 (0.43) MMP9MMP1ADAM17MMP3ADAM9
SCHEMBL7980335 0.85 ACE (0.48) F10POLBALDH1A1KDM4ECASP1
SCHEMBL7542044 0.80 PTPN1 (0.46) NR1D1POLBPTPN1
SCHEMBL11395371 0.77 NR1D1 (0.48) NR1D1POLBPTPN1
SCHEMBL11395379 0.77 NR1D1 (0.48) NR1D1POLBPTPN1
SCHEMBL5902094 0.76 FKBP1A (0.55) POLBALDH1A1HSD17B10SMN1; SMN2
SCHEMBL28557927 0.76 NR1D1 (0.67) MMP9MMP1ADAM17MMP3ADAM9
SCHEMBL29409300 0.76 NR1D1 (0.67) MMP9MMP1ADAM17MMP3ADAM9
SCHEMBL7976649 0.75 FKBP1A (0.53)
SCHEMBL7976654 0.75 FKBP1A (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6323215-B1 TREAT AND PREVENT DISORDERS CHARACTERIZED BY NEURONAL DAMAGE SUCH AS PARKINSON'S DISEASE, ALZHEIMER'S DISEASE, STROKE, MULTIPLE SCLEROSIS, AMYOTROPHIC LATERAL SCLEROSIS, DIABETIC NEUROPATHY AND BELL'S PALSY. ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-11-27 US disclosed