SCHEMBL7980335

SCHEMBL7980335

O=C(C(=O)N1Cc2ccccc2C[C@H]1C(=O)O)c1cccs1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.48
POLB P06746 3/20 0.45
TDP1 Q9NUW8 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CASP1 P29466 1/20 0.44
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
F10 P00742 1/20 0.42
SLC18A3 Q16572 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978564 0.85 MMP9 (0.43) POLBKDM4EALDH1A1CASP1CES2
SCHEMBL7978561 0.85 MMP9 (0.43) POLBKDM4EALDH1A1CASP1CES2
SCHEMBL7251696 0.77 CES2 (0.49) L3MBTL1KDM4EALDH1A1CES2CES1
SCHEMBL14397410 0.77 CES2 (0.49) L3MBTL1KDM4EALDH1A1CES2CES1
SCHEMBL14397408 0.76 ACE (0.59) ACEPOLBTDP1L3MBTL1
SCHEMBL4573235 0.76 ACE (0.61) ACEPOLBTDP1L3MBTL1KDM4E
SCHEMBL8908771 0.76 ACE (0.61) ACEPOLBTDP1L3MBTL1KDM4E
SCHEMBL3840630 0.76 ACE (0.61) ACEPOLBTDP1L3MBTL1KDM4E
SCHEMBL3149932 0.75 ALDH1A1 (0.48) POLBALDH1A1CES2CES1
SCHEMBL14407803 0.75 ALDH1A1 (0.48) POLBALDH1A1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6323215-B1 TREAT AND PREVENT DISORDERS CHARACTERIZED BY NEURONAL DAMAGE SUCH AS PARKINSON'S DISEASE, ALZHEIMER'S DISEASE, STROKE, MULTIPLE SCLEROSIS, AMYOTROPHIC LATERAL SCLEROSIS, DIABETIC NEUROPATHY AND BELL'S PALSY. ORTHO-MCNEIL PHARMACEUTICAL, INC. 2001-11-27 US disclosed