SCHEMBL7978741

SCHEMBL7978741

COc1ccccc1N1CCN(CCCCN2CSC3(CCCC3)C2=O)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.61
HTR7 P34969 3/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
DRD2 P14416 2/20 0.57
DRD3 P35462 2/20 0.57
DRD5 P21918 1/20 0.57
DRD1 P21728 1/20 0.56
DRD4 P21917 1/20 0.56
ADRA1B P35368 2/20 0.56
ALDH1A1 P00352 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
ALOX12 P18054 1/20 0.56
ADRA1D P25100 1/20 0.56
ADRA1A P35348 1/20 0.56
HIF1A Q16665 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9298422 0.99 HTR1A (0.60) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7991570 0.86 HTR1A (0.60) HTR1AHTR7MEN1KMT2ACYP1A2
Hydrochloric Acid SCHEMBL7990511 0.85 HTR1A (0.59) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7990156 0.79 HTR2A (0.51) HTR1ADRD2DRD4ADRA1A
SCHEMBL7990544 0.78 HTR7 (0.66) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL14761754 0.76 HTR1A (0.68) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7990516 0.76 HTR1A (0.60) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7996612 0.76 HTR1A (0.60) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7991154 0.76
SCHEMBL6526368 0.76 DRD2 (0.85) HTR1AHTR7MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037984-A Anticonvulsants; anxiolytic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US claimed
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed
US-5136037-A 3-(4-substituted-4-piperazinyl)butyl-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-08-04 US disclosed
US-5037984-A Anticonvulsants; anxiolytic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US disclosed
US-4933453-A ANTIPSYCHOTIC, ANALGESIC, ANTICONVULSANT, AND ANXIOLYTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-12 US disclosed