SCHEMBL7990516

SCHEMBL7990516

COc1ccccc1N1CCN(CCCCN2CS(=O)(=O)C(C)(C)C2=O)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.60
HTR7 P34969 6/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
DRD2 P14416 7/20 0.60
DRD3 P35462 5/20 0.60
DRD5 P21918 2/20 0.60
HTR6 P50406 3/20 0.59
ADRA1D P25100 2/20 0.59
ADRA1A P35348 2/20 0.59
ADRA1B P35368 2/20 0.59
ALDH1A1 P00352 2/20 0.59
TYR P14679 1/20 0.59
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
ALOX12 P18054 1/20 0.59
HIF1A Q16665 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991570 0.80 HTR1A (0.60) HTR1AHTR7MEN1KMT2ACYP1A2
Hydrochloric Acid SCHEMBL7990511 0.80 HTR1A (0.59) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7993118 0.80 HTR1A (0.62) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7989883 0.79 HTR1A (0.60) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL6526368 0.78 DRD2 (0.85) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7979558 0.76 HTR1A (0.62) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL13875119 0.76 HTR1A (1.00) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7978741 0.76 HTR1A (0.61) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL7990544 0.76 HTR7 (0.66) HTR1AHTR7MEN1KMT2ACYP1A2
SCHEMBL6017582 0.76 HTR7 (1.00) HTR1AHTR7MEN1KMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed