SCHEMBL7979012

SCHEMBL7979012

Cc1cc(C)c(-c2csc(C(=O)O)c2N)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
POLB P06746 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 1/20 0.38
DAO P14920 2/20 0.37
LMNA P02545 1/20 0.34
MYC P01106 1/20 0.33
TPMT P51580 1/20 0.33
GPR35 Q9HC97 2/20 0.33
LCK P06239 1/20 0.33
TTR P02766 1/20 0.33
PKM P14618 1/20 0.33
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CISD2 Q8N5K1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL535647 0.75 L3MBTL1 (0.52) KDM4EPOLBTDP1L3MBTL1ALDH1A1
Hydrochloric Acid SCHEMBL7034535 0.73 TDP1 (0.50) KDM4EPOLBTDP1L3MBTL1ALDH1A1
SCHEMBL10472839 0.73 L3MBTL1 (0.50) KDM4EPOLBTDP1L3MBTL1ALDH1A1
SCHEMBL6271882 0.70 ALDH1A1 (0.54) KDM4ETDP1ALDH1A1LMNAGPR35
SCHEMBL7609688 0.69 ALDH1A1 (0.33) KDM4EPOLBALDH1A1MAPT
SCHEMBL5154551 0.67 ALDH1A1 (0.49) KDM4EPOLBTDP1L3MBTL1ALDH1A1
SCHEMBL22068855 0.66 POLB (0.39) KDM4EPOLBTDP1L3MBTL1ALDH1A1
SCHEMBL5880332 0.66 HSD17B10 (0.52) KDM4EPOLBTDP1L3MBTL1ALDH1A1
SCHEMBL3459607 0.66 GPR35 (0.43) KDM4ETDP1ALDH1A1GPR35LCK
SCHEMBL27404772 0.66 POLB (0.42) KDM4EPOLBTDP1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211195-B1 NERVOUS SYSTEM, PSYCHOLOGICAL AND GLANDULAR DISORDERS NEUROCRINE BIOSCIENCES, INC. 2001-04-03 US disclosed
EP-0977759-A1 CRF ANTAGONISTIC THIOPHENOPYRIDINES JANSSEN PHARMACEUTICA N.V. (BE) 2000-02-09 EP disclosed
WO-1998047903-A1 CRF ANTAGONISTIC THIOPHENOPYRIDINES JANSSEN PHARMACEUTICA N.V. (BE) 1998-10-29 WO disclosed