SCHEMBL7979345

SCHEMBL7979345

CC1Oc2ccc(CN(Cc3cc(C(C)(C)C)c(O)c(C(C)(C)C)c3)C(=O)OC(C)(C)C)cc2N=C1N

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
TSHR P16473 1/20 0.34
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
RECQL P46063 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6302740 0.86 HDAC3 (0.43) GAAALDH1A1TSHRHDAC3HDAC1
SCHEMBL7978190 0.85 GAA (0.33) GAAALDH1A1LMNATSHRHDAC3
SCHEMBL6303033 0.84 L3MBTL1 (0.37) GAAHDAC3HDAC1HDAC2NCOR2
SCHEMBL6310829 0.84 RIPK1 (0.36) TSHRHDAC3HDAC1HDAC2NCOR2
SCHEMBL6302989 0.83 HDAC3 (0.35) TSHRHDAC3HDAC1HDAC2NCOR2
SCHEMBL6608622 0.83 GAA (0.32) GAAHDAC3HDAC1HDAC2NCOR2
SCHEMBL5189245 0.83 SSTR4 (0.32) HDAC3HDAC1HDAC2NCOR2
SCHEMBL5188660 0.83 SSTR4 (0.32) HDAC3HDAC1HDAC2NCOR2
SCHEMBL6303012 0.82 HDAC3 (0.31) HDAC3HDAC1HDAC2NCOR2
SCHEMBL6302903 0.81 NR1D1 (0.37) ALDH1A1LMNAHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001081324-A1 BENZOXAZINE DERIVATIVES AND BENZOTHIAZINE DERIVATIVES HAVING NOS-INHIBITORY AND ANTIOXIDANT PROPERTIES SCHERING AKTIENGESELLSCHAFT (DE) 2001-11-01 WO disclosed