SCHEMBL7982616

SCHEMBL7982616

CC(=O)Nc1oc(-c2cccc(-c3ccc(-c4ccc5ccccc5c4)cc3)c2O)nc1-c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.56
FLT1 P17948 1/20 0.56
FLT4 P35916 1/20 0.56
SIRT2 Q8IXJ6 4/20 0.44
CYP19A1 P11511 3/20 0.43
CYP11B1 P15538 3/20 0.43
CYP11B2 P19099 3/20 0.43
CYP17A1 P05093 1/20 0.43
CCNE2 O96020 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
ALOX15 P16050 1/20 0.40
PIK3CA P42336 1/20 0.39
PIK3CG P48736 1/20 0.39
UTRN P46939 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ABL1 P00519 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980265 0.89 SIRT2 (0.52) KDRFLT1FLT4SIRT2CYP19A1
SCHEMBL7979621 0.88 KDR (0.50) KDRFLT1FLT4CCNE2CCNE1
SCHEMBL7969453 0.87 HPGD (0.46) KDRFLT1FLT4SIRT2CYP19A1
SCHEMBL7980821 0.87 KDR (0.54) KDRFLT1FLT4CYP19A1CCNE2
SCHEMBL7983601 0.87 KDR (0.53) KDRFLT1FLT4CCNE2CCNE1
SCHEMBL7983236 0.85 KDR (0.54) KDRFLT1FLT4CCNE2CCNE1
SCHEMBL7739014 0.84 KDR (0.63) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7979692 0.84 KDR (0.54) KDRFLT1FLT4ALOX15PIK3CA
SCHEMBL7979899 0.83 KDR (0.52) KDRFLT1FLT4SIRT2CCNE2
SCHEMBL7739016 0.81 KDR (0.56) KDRFLT1FLT4CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed