SCHEMBL7982908

SCHEMBL7982908

CC(Br)C(=O)CC(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.52
ALDH1A1 P00352 3/20 0.52
MAPT P10636 1/20 0.52
GAA P10253 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.50
MAPK1 P28482 1/20 0.50
RAB9A P51151 2/20 0.47
HTT P42858 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1555636 0.84 ALDH1A1 (0.59) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL7892509 0.84 GAA (0.54) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL7903564 0.83 ALDH1A1 (0.51) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL7905669 0.82 HTR2A (0.56) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL27787118 0.81 GAA (0.60) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL5765803 0.81 ALDH1A1 (0.57) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL11094410 0.81 ALDH1A1 (0.56) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL9344653 0.80 LMNA (0.57) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL1554845 0.80 ALDH1A1 (0.55) HTR2AALDH1A1MAPTGAAL3MBTL1
SCHEMBL5724425 0.80 ALDH1A1 (0.59) HTR2AALDH1A1MAPTGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed