SCHEMBL7983285

SCHEMBL7983285

Oc1cc2c(cc1O)-c1cc(O)c(O)cc1C2=Cc1ccccc1C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.44
TNF P01375 2/20 0.43
IL6 P05231 2/20 0.43
GRIN2D O15399 2/20 0.41
GRIN3B O60391 2/20 0.41
GRIN1 Q05586 2/20 0.41
GRIN2A Q12879 2/20 0.41
GRIN2B Q13224 2/20 0.41
GRIN2C Q14957 2/20 0.41
GRIN3A Q8TCU5 2/20 0.41
MAOB P27338 4/20 0.40
P4HB P07237 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
MYC P01106 1/20 0.38
MAX P61244 1/20 0.38
CYP24A1 Q07973 1/20 0.38
BAX Q07812 2/20 0.38
MAOA P21397 1/20 0.38
BACE1 P56817 1/20 0.38
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9372017 0.80 TNF (0.46) TNFIL6MAOBCYP24A1MAPT
SCHEMBL4157687 0.73 TNF (0.50) NFKB1TNFIL6GRIN2DGRIN3B
SCHEMBL7983283 0.69 NQO2 (0.54)
SCHEMBL7980865 0.69 LCK (0.46) BACE1MAPT
SCHEMBL29446986 0.68 NFKB1 (0.52) NFKB1TNFIL6GRIN2DGRIN3B
SCHEMBL165004 0.68 NFKB1 (0.52) NFKB1TNFIL6GRIN2DGRIN3B
SCHEMBL11126093 0.68 NFKB1 (0.57) NFKB1TNFIL6GRIN2DGRIN3B
SCHEMBL25375799 0.67 TNF (0.59) NFKB1TNFIL6GRIN2DGRIN3B
SCHEMBL2494559 0.67 NFKB1 (0.55) NFKB1TNFIL6GRIN2DGRIN3B
SCHEMBL323188 0.65 NFKB1 (0.53) NFKB1TNFIL6GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194439-B1 ANTICANCER AGENT PFIZER INC. 2001-02-27 US disclosed
EP-0586608-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1994-03-16 EP disclosed
WO-1992021660-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER, INC. (US) 1992-12-10 WO disclosed