SCHEMBL7985338

SCHEMBL7985338

CC(=O)N(c1ccccc1)c1ccccc1C

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
TSHR P16473 1/20 0.54
NPSR1 Q6W5P4 4/20 0.48
LMNA P02545 2/20 0.47
ALDH1A1 P00352 3/20 0.46
NPC1 O15118 3/20 0.45
APAF1 O14727 1/20 0.45
TRPM8 Q7Z2W7 2/20 0.42
RAB9A P51151 2/20 0.41
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22917037 0.88 LMNA (0.53) KMT2AMEN1TSHRNPSR1LMNA
SCHEMBL2092543 0.86 TRPM8 (0.51) KMT2AMEN1TSHRNPSR1LMNA
SCHEMBL2719421 0.86 LMNA (0.48) KMT2AMEN1TSHRNPSR1LMNA
SCHEMBL2092538 0.85 NPSR1 (0.48) KMT2AMEN1TSHRNPSR1LMNA
SCHEMBL22917197 0.84 HSD17B1 (0.45) KMT2AMEN1TSHRLMNAALDH1A1
SCHEMBL11613737 0.83 NPSR1 (0.47) KMT2AMEN1TSHRNPSR1LMNA
SCHEMBL15999740 0.81 NR3C2 (0.49) KMT2AMEN1TSHRNPSR1ALDH1A1
SCHEMBL741752 0.81 NPSR1 (0.64) KMT2AMEN1TSHRNPSR1ALDH1A1
SCHEMBL17472225 0.81 SIGMAR1 (0.42) KMT2AMEN1TSHRNPSR1LMNA
SCHEMBL8779541 0.79 TRPM8 (0.51) KMT2AMEN1TSHRNPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103102303-B As the benzyl amine derivative of CETP inhibitor DR. REDDY'S LABORATORIES LTD. (IN) 2015-10-28 CN disclosed
CN-103102303-A Benzylamine derivatives as CETP inhibitors REDDY US THERAPEUTICS INC 2013-05-15 CN disclosed
CN-101443006-B Novel benzylamine derivatives as CETP inhibitors REDDY US THERAPEUTICS INC 2012-10-10 CN disclosed
CN-101443006-A Novel benzylamine derivatives as CETP inhibitors REDDY US THERAPEUTICS INC (US) 2009-05-27 CN disclosed
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP disclosed