1,2,3-Benzothia-Diazole-7-Carboxylic Acid

1,2,3-Benzothia-Diazole-7-Carboxylic Acid

SCHEMBL7986261

CCC(C)NN.O=C(O)c1cccc2nnsc12

nearest known ligand 0.36

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
KDM4E B2RXH2 4/20 0.34
MAPT P10636 3/20 0.34
HTT P42858 1/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
ALDH1A1 P00352 3/20 0.33
TP53 P04637 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
RAB9A P51151 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NPC1 O15118 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
ASPH Q12797 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1,2,3-Benzothia-Diazole-7-Carboxylic Acid SCHEMBL2455715 0.82 ALDH1A1 (0.44) KMT2AMEN1KDM4EMAPTHTT
SCHEMBL9668606 0.81 MEN1 (0.40) KMT2AMEN1KDM4EMAPTHTT
1,2,3-Benzothia-Diazole-7-Carboxylic Acid SCHEMBL9084433 0.81 ALDH1A1 (0.43) KMT2AMEN1KDM4EMAPTHTT
1,2,3-Benzothia-Diazole-7-Carboxylic Acid SCHEMBL8588144 0.78 MAPT (0.45) KMT2AMEN1KDM4EMAPTGAA
SCHEMBL7986259 0.77 MAPT (0.34) KMT2AKDM4EMAPTGAALMNA
SCHEMBL4031502 0.77 GAA (0.44) KMT2AMEN1KDM4EMAPTGAA
SCHEMBL9088391 0.75 ADRA1A (0.41) KMT2AMEN1KDM4EMAPTGAA
SCHEMBL3743917 0.75 ATM (0.32) KMT2AMEN1KDM4EMAPTHTT
SCHEMBL8051642 0.72 MAPT (0.45) KMT2AMEN1MAPTLMNAALDH1A1
SCHEMBL3743974 0.72 PARP1 (0.40) KMT2AMEN1KDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6262342-B1 CHEMICALLY REGULATABLE DNA SEQUENCES DERIVED FROM 5' REGION OF GENES ENCODING PATHOGENESIS RELATED PROTEINS CAPABLE OF REGULATING TRANSCRIPTION OF AN ASSOCIATED DNA SEQUENCE IN PLANTS/TISSUES, CHIMERIC CONSTRUCTS, AND TRANSGENIC PLANTS NOVARTIS FINANCE CORPORATION 2001-07-17 US disclosed
US-5880328-A ANTI-PATHOGENIC SEQUENCES DERIVED FROM NOVEL CDNAS CODING FOR PR PROTEINS WHICH CAN BE GENETICALLY ENGINEERED AND TRANSFORMED INTO PLANTS TO CONFER ENHANCED RESISTANCE TO DISEASE NOVARTIS FINANCE CORPORATION (US) 1999-03-09 US disclosed
US-5847258-A DNA encoding β-1,3-glucanases NOVARTIS FINANCE CORPORATION (US) 1998-12-08 US disclosed