SCHEMBL793623

SCHEMBL793623

COc1cc2c(cc1Cl)CN(c1cnccc1C)CC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.52
ALDH1A1 P00352 3/20 0.52
LMNA P02545 3/20 0.52
MAPK1 P28482 2/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MAOB P27338 4/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
GAA P10253 2/20 0.42
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.40
CYP1A2 P05177 1/20 0.40
HTR2C P28335 1/20 0.40
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
ACHE P22303 1/20 0.39
PDE4B Q07343 1/20 0.39
MAOA P21397 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL798146 0.83 DRD1 (0.42) MAPTALDH1A1LMNAMAPK1HTT
SCHEMBL793474 0.83 CYP11B2 (0.41) MAPTALDH1A1LMNAMAPK1HTT
SCHEMBL798533 0.80 TIPARP (0.46) MAPTALDH1A1
SCHEMBL798654 0.77 PDGFRB (0.43)
SCHEMBL794032 0.76 CYP11B2 (0.44) MAPTALDH1A1LMNAMAPK1HTT
SCHEMBL798675 0.76 TIPARP (0.46) MAPTALDH1A1LMNAHPGDACHE
SCHEMBL793143 0.74 GRIN2D (0.42) MAPTALDH1A1KMT2AMEN1GAA
SCHEMBL794272 0.71 PHGDH (0.43) HTR2C
SCHEMBL793875 0.71 TRPV3 (0.41) HTR2C
SCHEMBL26955904 0.70 MAOA (0.77) MAPTALDH1A1LMNAMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP disclosed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO disclosed