SCHEMBL7987433

SCHEMBL7987433

COc1cccc(Cn2cnc3nc(-c4cccnc4)nc(O)c32)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.54
MAPT P10636 2/20 0.46
GAA P10253 1/20 0.45
TP53 P04637 2/20 0.44
RXFP1 Q9HBX9 1/20 0.44
TNIK Q9UKE5 2/20 0.44
ROCK1 Q13464 2/20 0.43
CYP19A1 P11511 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
ABCB1 P08183 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7985850 0.90 GAA (0.49) ROCK2GAATP53RXFP1ROCK1
SCHEMBL7989313 0.89 ROCK2 (0.52) ROCK2GAATP53RXFP1ROCK1
SCHEMBL7974018 0.89 GAA (0.53) ROCK2MAPTGAATP53RXFP1
SCHEMBL7988934 0.87 CYP1A2 (0.47) ROCK2MAPTCYP1A2CYP3A4CYP2D6
SCHEMBL7984696 0.87 GAA (0.47) ROCK2GAATP53RXFP1ROCK1
SCHEMBL7985653 0.86 GAA (0.46) ROCK2GAATP53RXFP1ROCK1
SCHEMBL7974093 0.85 GAA (0.48) ROCK2MAPTGAATP53RXFP1
SCHEMBL7974314 0.85 GAA (0.46) ROCK2GAATP53RXFP1ROCK1
SCHEMBL7988659 0.85 P2RX7 (0.41) MAPTCYP3A4CYP2D6CYP2C19ABCG2
SCHEMBL7985334 0.85 ABCG2 (0.46) ALDH1A1ABCG2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6310070-B1 FOR TREATING NEPHRITIS, IMPROVING PROTEINURIA DUE TO GLOMERULONEPHRITIS AND PREVENTING AGGRAVATION OF NEPHRITIS JAPAN ENERGY CORPORATION (JP) 2001-10-30 US disclosed
EP-0999211-A1 NOVEL PURINE DERIVATIVES AND MEDICINAL USE THEREOF JAPAN ENERGY CORPORATION (JP) 2000-05-10 EP disclosed