SCHEMBL7993934

SCHEMBL7993934

COc1cccc2c(-c3cncc(-c4ccsc4)c3)cn(CCCN3CCCCC3)c12

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.70
FLT1 P17948 4/20 0.70
FLT4 P35916 4/20 0.70
CNR2 P34972 2/20 0.44
DRD2 P14416 5/20 0.40
DRD3 P35462 5/20 0.40
DRD4 P21917 4/20 0.40
HTR1A P08908 4/20 0.40
GSK3B P49841 4/20 0.39
QPCT Q16769 2/20 0.39
SLC6A2 P23975 1/20 0.37
HTR2A P28223 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
NFATC1 O95644 1/20 0.37
DYRK1A Q13627 1/20 0.37
KCNH2 Q12809 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990673 0.95 KDR (0.69) KDRFLT1FLT4CNR2DRD2
SCHEMBL7554218 0.94 KDR (0.71) KDRFLT1FLT4CNR2DRD2
SCHEMBL7550389 0.88 KDR (0.55) KDRFLT1FLT4CNR2DRD2
SCHEMBL7987725 0.87 KDR (0.70) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7549404 0.87 KDR (0.51) KDRFLT1FLT4CNR2DRD2
SCHEMBL7554716 0.86 KDR (0.51) KDRFLT1FLT4CNR2DRD2
SCHEMBL7555367 0.86 KDR (0.51) KDRFLT1FLT4CNR2GSK3B
SCHEMBL7553648 0.85 KDR (0.50) KDRFLT1FLT4CNR2DRD2
SCHEMBL7990971 0.85 KDR (0.70) KDRFLT1FLT4CNR2
SCHEMBL7556349 0.83 KDR (0.58) KDRFLT1FLT4CNR2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed