SCHEMBL7987979

SCHEMBL7987979

COC(=O)CCCCOc1ccc2c(c1)CCN=C2C(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.46
S1PR1 P21453 5/20 0.43
LTA4H P09960 1/20 0.42
PDE3B Q13370 3/20 0.40
PDE3A Q14432 3/20 0.40
P2RY12 Q9H244 3/20 0.40
LTB4R Q15722 1/20 0.40
PDE2A O00408 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
LSS P48449 1/20 0.38
S1PR3 Q99500 2/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7989163 0.88 PTPN11 (0.48) PPARALMNAMAPK1L3MBTL1CA1
SCHEMBL7995609 0.84 S1PR1 (0.40) PPARAS1PR1KDM4ESMN1; SMN2LSS
SCHEMBL7994778 0.81 SLC2A1 (0.41) PPARAS1PR1KDM4ENPC1MAPT
SCHEMBL7987543 0.80 ABCB1 (0.44) S1PR1KDM4EMAPTSMN1; SMN2S1PR3
SCHEMBL7994780 0.80 MAOB (0.53) S1PR1KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL7988818 0.78 MAOB (0.48) NPC1MAPTRAB9ASMN1; SMN2MAPK1
SCHEMBL7991609 0.75 MAOB (0.49) NPC1RAB9ASMN1; SMN2L3MBTL1MAOA
SCHEMBL7991453 0.73 KDM4E (0.51) KDM4EMAPTMAPK1MAOA
SCHEMBL7989235 0.73 ACHE (0.48) KDM4ENPC1MAPTRAB9ASMN1; SMN2
SCHEMBL7991147 0.70 MAOB (0.47) S1PR1KDM4ENPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed