SCHEMBL7989050

SCHEMBL7989050

COc1ccc(-c2ccc(C(=O)O)c(-c3cccc(Cl)c3)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.52
AKR1C2 P52895 1/20 0.52
DCLRE1B Q9H816 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
LMNA P02545 1/20 0.50
HPGD P15428 1/20 0.50
GFER P55789 1/20 0.50
PKM P14618 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ACLY P53396 1/20 0.46
GRIK1 P39086 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
SLC6A9 P48067 1/20 0.46
PRKAB2 O43741 2/20 0.46
PRKAG1 P54619 2/20 0.46
PRKAA2 P54646 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16527361 0.83 SMN1; SMN2 (0.62) AKR1C3AKR1C2SMN1; SMN2MEN1KMT2A
SCHEMBL30996183 0.81 ABL1 (0.63) KMT2AHDAC4HDAC2HDAC8
SCHEMBL8480988 0.81 ABL1 (0.63) KMT2AHDAC4HDAC2HDAC8
SCHEMBL8202718 0.79 PRKAB2 (0.55) AKR1C3AKR1C2SMN1; SMN2LMNAHPGD
SCHEMBL7591657 0.77 SMN1; SMN2 (0.75) AKR1C3AKR1C2SMN1; SMN2HPGDPRKAB2
SCHEMBL7553675 0.76 RARA (0.58) ACLYSLC6A9MAP4K4
SCHEMBL27542071 0.76 BACE1 (0.56) SMN1; SMN2MEN1KMT2AHPGDHDAC4
SCHEMBL28694686 0.76 DCLRE1B (0.56) AKR1C2DCLRE1BACLYGRIK1MAP4K4
SCHEMBL7606419 0.75 PTPN11 (0.53) SMN1; SMN2HPGDNPC1RAB9AKDM4E
SCHEMBL6701301 0.75 SMN1; SMN2 (0.63) AKR1C3AKR1C2SMN1; SMN2LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6258843-B1 DRUGS AS ENZYME INHIBITORS NOVARTIS AG (CH) 2001-07-10 US disclosed