SCHEMBL7989895

SCHEMBL7989895

O=C(O)c1nc(-c2ccc(N3CCCCCC3)cc2)[nH]c1-c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.50
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
TP53 P04637 2/20 0.47
MAPK1 P28482 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MAPK13 O15264 1/20 0.45
ALOX5 P09917 1/20 0.45
TGFBR1 P36897 1/20 0.45
MAPK12 P53778 1/20 0.45
MAPK11 Q15759 1/20 0.45
MAPK14 Q16539 1/20 0.45
SIRT2 Q8IXJ6 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7977819 0.99 CHEK2 (0.51) CHEK2NPC1RAB9ATP53MAPK1
SCHEMBL7991747 0.89 PARP1 (0.53) CHEK2ALDH1A1MAPTKDM4EMAPK13
SCHEMBL7989662 0.88 LMNA (0.45) CHEK2ALDH1A1MAPTHPGDSIRT2
SCHEMBL7989265 0.87 SIRT2 (0.47) CHEK2NPC1RAB9ATP53ALDH1A1
SCHEMBL7991843 0.87 AURKA (0.45) CHEK2ALDH1A1MAPTHPGDSIRT2
SCHEMBL7978031 0.84 SIRT2 (0.61) CHEK2NPC1RAB9ATP53ALDH1A1
SCHEMBL7977935 0.84 CHEK2 (0.53) CHEK2RAB9ATP53ALDH1A1MAPT
SCHEMBL7987913 0.82 SIRT2 (0.59) CHEK2NPC1RAB9ATP53MAPK1
SCHEMBL7989851 0.82 PARP1 (0.45) CHEK2ALDH1A1MAPTKDM4EHPGD
SCHEMBL7988176 0.79 ALDH1A1 (0.44) CHEK2NPC1RAB9ATP53MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288061-B1 INTERLEUKIN INHIBITORS; ASTHMA, BRONCHODILATOR AGENTS, ANTIALLERGENS WELFIDE CORPORATION (JP) 2001-09-11 US disclosed