SCHEMBL7991747

SCHEMBL7991747

O=C(O)c1nc(-c2ccc(N3CCOCC3)cc2)[nH]c1-c1ccc(F)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.53
CHEK2 O96017 1/20 0.49
PIN1 Q13526 1/20 0.46
CFTR P13569 1/20 0.46
AKR1C3 P42330 1/20 0.46
PRKAB2 O43741 1/20 0.46
PRKAG1 P54619 1/20 0.46
PRKAA2 P54646 1/20 0.46
PRKAA1 Q13131 1/20 0.46
PRKAG3 Q9UGI9 1/20 0.46
PRKAG2 Q9UGJ0 1/20 0.46
PRKAB1 Q9Y478 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
ALOX5 P09917 2/20 0.45
MAPK13 O15264 1/20 0.44
TGFBR1 P36897 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7977819 0.91 CHEK2 (0.51) PARP1CHEK2SIRT2SIRT1ALOX5
SCHEMBL7989851 0.90 PARP1 (0.45) PARP1CHEK2PIN1CFTRAKR1C3
SCHEMBL7989895 0.89 CHEK2 (0.50) PARP1CHEK2SIRT2SIRT1ALOX5
SCHEMBL7991773 0.88 PARP1 (0.51) PARP1CHEK2PIN1AKR1C3PRKAB2
SCHEMBL7989978 0.84 SIRT2 (0.61) PARP1CHEK2SIRT2SIRT1ALOX5
SCHEMBL7989922 0.81 SIRT2 (0.48) PARP1CHEK2PIN1CFTRPRKAB2
SCHEMBL7978052 0.80 PARP1 (0.46) PARP1MEN1KMT2AGAAMAPT
SCHEMBL7991959 0.79 SMN1; SMN2 (0.44) PARP1PIN1AKR1C3PRKAB2PRKAG1
SCHEMBL7989265 0.79 SIRT2 (0.47) CHEK2PIN1SIRT2SIRT1MEN1
SCHEMBL7991843 0.79 AURKA (0.45) PARP1CHEK2AKR1C3PRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288061-B1 INTERLEUKIN INHIBITORS; ASTHMA, BRONCHODILATOR AGENTS, ANTIALLERGENS WELFIDE CORPORATION (JP) 2001-09-11 US disclosed