SCHEMBL7990111

SCHEMBL7990111

COc1cccc(C(CC[N])CCCc2cccnc2)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 10/20 0.49
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
KDM4E B2RXH2 1/20 0.42
GFER P55789 1/20 0.42
PTGDR Q13258 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KCNA5 P22460 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159742 0.89 PTAFR (0.49) PTAFRHTR1ADRD2KDM4EGFER
SCHEMBL6165461 0.75 ALDH1A1 (0.55) PTAFRALDH1A1
SCHEMBL28177088 0.74 HTR1A (0.67) PTAFRHTR1ADRD2KDM4EGFER
SCHEMBL6160650 0.73 CYP2A6 (0.51) PTAFR
SCHEMBL6159739 0.72 CHRM2 (0.56) PTAFRHTR1ADRD2PTGDRTDP1
SCHEMBL6158970 0.70 CYP2A6 (0.48) PTAFRKDM4EALDH1A1HTTTDP1
SCHEMBL3344537 0.70 CASR (0.71) ALDH1A1LMNAHTT
SCHEMBL2462030 0.70 CASR (0.71) ALDH1A1LMNAHTT
SCHEMBL11486476 0.69 ROCK1 (0.44)
SCHEMBL28705794 0.69 TDP1 (0.57) TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228872-B1 PEPTIDE-PROLYL ISOMERASE AND ROTAMASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY 2001-05-08 US disclosed