SCHEMBL7992026

SCHEMBL7992026

CCOC(=O)Cc1cc2c(s1)CCN(C(=O)[C@H](Cc1ccc([N+](=O)[O-])cc1)NC(=O)CCC1CCNCC1)C2.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.35

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.35
ITGA2B P08514 9/20 0.35
ITGA4 P13612 1/20 0.33
P2RX7 Q99572 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MCL1 Q07820 2/20 0.33
ADORA1 P30542 1/20 0.32
MMP2 P08253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974860 0.85 YAP1 (0.40) ITGB3ITGA2BITGA4P2RX7KMT2A
Hydrochloric Acid SCHEMBL7986192 0.84 ITGB3 (0.39) ITGB3ITGA2BP2RX7MEN1KMT2A
Trifluoroacetic Acid SCHEMBL7992078 0.81 ITGB3 (0.35) ITGB3ITGA2BP2RX7KMT2AADORA1
SCHEMBL7985559 0.80 ADORA1 (0.50) ITGB3ITGA2BITGA4P2RX7KMT2A
SCHEMBL7992105 0.77 YAP1 (0.41) ITGB3ITGA2BITGA4KMT2AMCL1
SCHEMBL7986612 0.77 ITGB3 (0.40) ITGB3ITGA2BP2RX7KMT2AMCL1
SCHEMBL7988424 0.77 ITGB3 (0.57) ITGB3ITGA2BP2RX7MEN1KMT2A
Hydrochloric Acid SCHEMBL7986317 0.76 ITGB3 (0.56) ITGB3ITGA2BP2RX7MEN1KMT2A
SCHEMBL7992407 0.76 ITGB3 (0.48) ITGB3ITGA2BP2RX7MEN1KMT2A
SCHEMBL7986354 0.76 ITGB3 (0.47) ITGB3ITGA2BP2RX7MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265418-B1 ANTICOAGULANTS UBE INDUSTRIES, LTD. (JP) 2001-07-24 US disclosed
EP-1020467-A1 N-ACYLAMINO ACID AMIDE COMPOUNDS AND INTERMEDIATES FOR PREPARATION THEREOF UBE INDUSTRIES LIMITED (JP) 2000-07-19 EP disclosed