SCHEMBL7993018

SCHEMBL7993018

COc1cc2c(N)cc(-c3nc(C(C)C)cs3)nc2cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.41
GAA P10253 1/20 0.35
NPC1 O15118 1/20 0.35
P2RX3 P56373 1/20 0.34
P2RX2 Q9UBL9 1/20 0.34
HSP90AA1 P07900 2/20 0.33
HSP90AB1 P08238 2/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
PGK1 P00558 3/20 0.32
GSK3B P49841 1/20 0.32
MAP4K2 Q12851 1/20 0.32
THRB P10828 1/20 0.31
BLM P54132 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ADRA1D P25100 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL314417 0.86 PDE3B (0.33) GAANPC1PDE3BPDE3AALDH1A1
SCHEMBL8003339 0.82 POLB (0.39) GAAP2RX3P2RX2PDE3BPDE3A
SCHEMBL15216079 0.81 SLC2A1 (0.40) SLC2A1GAANPC1KDM4EALDH1A1
SCHEMBL8005887 0.81 SLC2A1 (0.40) SLC2A1GAANPC1HSP90AA1HSP90AB1
SCHEMBL15216087 0.81 SLC2A1 (0.42) SLC2A1GAANPC1P2RX3P2RX2
SCHEMBL15216084 0.79 ACHE (0.40) SLC2A1GAANPC1KDM4EALDH1A1
SCHEMBL8004279 0.79 SHMT1 (0.31)
SCHEMBL8006162 0.79 ALDH1A1 (0.37) SLC2A1NPC1KDM4EALDH1A1SMN1; SMN2
SCHEMBL577763 0.77 PGK1 (0.32) PGK1GSK3BMAP4K2APLNR
SCHEMBL15216076 0.77 CYP1A1 (0.35) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250174-B1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2013-08-28 EP disclosed
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed