SCHEMBL7993153

SCHEMBL7993153

CNS(=O)(=O)c1ccc(Oc2ccc(C)cn2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.60
LMNA P02545 3/20 0.60
HTT P42858 2/20 0.60
GAA P10253 2/20 0.54
ALDH1A1 P00352 4/20 0.51
KDM4E B2RXH2 3/20 0.49
IDO1 P14902 1/20 0.47
FFAR1 O14842 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
ADAMTS4 O75173 1/20 0.42
MMP1 P03956 1/20 0.42
MMP2 P08253 1/20 0.42
MMP13 P45452 1/20 0.42
MMP14 P50281 1/20 0.42
ADAMTS5 Q9UNA0 1/20 0.42
USP2 O75604 1/20 0.42
PTGS1 P23219 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402420 0.87 ALDH1A1 (0.51) SMN1; SMN2LMNAHTTGAAALDH1A1
SCHEMBL972533 0.83 KDM4E (0.53) SMN1; SMN2LMNAHTTGAAALDH1A1
SCHEMBL7994583 0.83 PTGS2 (0.56) SMN1; SMN2LMNAHTTGAAALDH1A1
SCHEMBL973305 0.82 ALDH1A1 (0.55) LMNAHTTGAAALDH1A1KDM4E
SCHEMBL8736878 0.81 SMN1; SMN2 (0.85) SMN1; SMN2LMNAHTTGAAALDH1A1
SCHEMBL20988347 0.81 IDO1 (0.63) SMN1; SMN2LMNAHTTALDH1A1IDO1
SCHEMBL13876057 0.81 LMNA (0.54) SMN1; SMN2LMNAHTTALDH1A1IDO1
SCHEMBL10153980 0.81 ADAMTS4 (0.62) SMN1; SMN2LMNAHTTALDH1A1KDM4E
Ammonia Solution, Strong SCHEMBL3402419 0.81 ALDH1A1 (0.53) LMNAHTTGAAALDH1A1KDM4E
SCHEMBL8737052 0.79 KDM4E (0.66) SMN1; SMN2HTTGAAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005783-A1 PYRROLIDINYL AND PIPERIDINYL COMPOUNDS USEFUL AS NHE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-14 WO disclosed