SCHEMBL7994923

SCHEMBL7994923

COc1cccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4ccc(Cl)cc34)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 1/20 0.40
GSK3B P49841 1/20 0.40
HTR6 P50406 2/20 0.36
CCNT1 O60563 1/20 0.36
CCNE1 P24864 1/20 0.36
CDK2 P24941 1/20 0.36
CDK7 P50613 1/20 0.36
CDK9 P50750 1/20 0.36
CCNH P51946 1/20 0.36
MNAT1 P51948 1/20 0.36
CYP2C19 P33261 1/20 0.35
CHEK1 O14757 2/20 0.35
EED O75530 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4D Q08499 1/20 0.34
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
SRC P12931 1/20 0.34
ABL2 P42684 1/20 0.34
CYP11B1 P15538 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990984 0.94 CCNT1 (0.36) PRKCAGSK3BHTR6CCNT1CCNE1
SCHEMBL7993914 0.94 HTR6 (0.38) PRKCAGSK3BHTR6CCNT1CCNE1
SCHEMBL7975970 0.93 HTR6 (0.39) HTR6CYP2C19CHEK1EEDPDE4B
SCHEMBL7503926 0.92 CCNT1 (0.38) HTR6CCNT1CCNE1CDK2CDK7
SCHEMBL7976151 0.91 CCNT1 (0.37) HTR6CCNT1CCNE1CDK2CDK7
SCHEMBL7976272 0.90 CCNT1 (0.41) PRKCAGSK3BHTR6CCNT1CCNE1
SCHEMBL7990169 0.89 PDE4B (0.37) HTR6CCNT1CCNE1CDK2CDK7
SCHEMBL7987305 0.89 CCNT1 (0.42) HTR6CCNT1CCNE1CDK2CDK7
SCHEMBL7990463 0.89 CHEK1 (0.39) CYP2C19CHEK1EEDACP1
SCHEMBL7990448 0.88 CYP11B1 (0.40) HTR6CCNT1CCNE1CDK2CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed