SCHEMBL7976272

SCHEMBL7976272

COc1cccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4ccccc34)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
CDK7 P50613 1/20 0.41
CDK9 P50750 1/20 0.41
CCNH P51946 1/20 0.41
MNAT1 P51948 1/20 0.41
ACP1 P24666 1/20 0.39
CYP2C19 P33261 1/20 0.37
CHEK1 O14757 2/20 0.37
PRKCA P17252 1/20 0.36
GSK3B P49841 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7975970 0.93 HTR6 (0.39) ACP1CYP2C19CHEK1LMNACYP1A2
SCHEMBL7986667 0.91 CDK7 (0.44) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7994923 0.90 PRKCA (0.40) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7990984 0.90 CCNT1 (0.36) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7987981 0.90 EGFR (0.38) ACP1CYP2C19CHEK1ALDH1A1LMNA
SCHEMBL7513288 0.89 CDK7 (0.47) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7990448 0.89 CYP11B1 (0.40) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7990463 0.89 CHEK1 (0.39) ACP1CYP2C19CHEK1EED
SCHEMBL7991127 0.88 CDK7 (0.46) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7990422 0.87 ABL1 (0.38) CCNT1CCNE1CDK2CDK7CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed