SCHEMBL7990448

SCHEMBL7990448

COc1ccc2c(c1)c(-c1cncc(-c3ccccc3)c1)cn2C(C)C1CCCNC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PDE4B Q07343 2/20 0.38
PDE4D Q08499 2/20 0.38
HTR6 P50406 4/20 0.38
CCNT1 O60563 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK7 P50613 1/20 0.38
CDK9 P50750 1/20 0.38
CCNH P51946 1/20 0.38
MNAT1 P51948 1/20 0.38
CASR P41180 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
DRD3 P35462 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987194 0.95 HTR6 (0.37) CYP11B1CYP11B2PDE4BPDE4DHTR6
SCHEMBL7975970 0.94 HTR6 (0.39) CYP11B1CYP11B2PDE4BPDE4DHTR6
SCHEMBL7990169 0.91 PDE4B (0.37) CYP11B1CYP11B2PDE4BPDE4DHTR6
SCHEMBL7993914 0.91 HTR6 (0.38) CYP11B1CYP11B2PDE4BPDE4DHTR6
SCHEMBL7986667 0.90 CDK7 (0.44) CYP11B1CYP11B2HTR6CCNT1CCNE1
SCHEMBL7976272 0.89 CCNT1 (0.41) CYP11B1CYP11B2HTR6CCNT1CCNE1
SCHEMBL7976003 0.88 PRKCZ (0.40) PDE4BPDE4DHTR6CDK2PRKCZ
SCHEMBL7513288 0.88 CDK7 (0.47) CCNT1CCNE1CDK2CDK7CDK9
SCHEMBL7976151 0.88 CCNT1 (0.37) PDE4BPDE4DHTR6CCNT1CCNE1
SCHEMBL7987305 0.88 CCNT1 (0.42) HTR6CCNT1CCNE1CDK2CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed