SCHEMBL7975970

SCHEMBL7975970

COc1cccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4ccc(OC)cc34)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.39
CYP2C19 P33261 2/20 0.37
CHEK1 O14757 2/20 0.37
EED O75530 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4D Q08499 1/20 0.36
EGFR P00533 2/20 0.36
ABL1 P00519 1/20 0.36
SRC P12931 1/20 0.36
ABL2 P42684 1/20 0.36
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
ACP1 P24666 1/20 0.35
AXL P30530 1/20 0.35
FLT3 P36888 1/20 0.35
TYRO3 Q06418 1/20 0.35
MERTK Q12866 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990448 0.94 CYP11B1 (0.40) HTR6PDE4BPDE4DCYP11B1CYP11B2
SCHEMBL7994923 0.93 PRKCA (0.40) HTR6CYP2C19CHEK1EEDPDE4B
SCHEMBL7993914 0.93 HTR6 (0.38) HTR6EEDPDE4BPDE4DEGFR
SCHEMBL7976272 0.93 CCNT1 (0.41) HTR6CYP2C19CHEK1EEDEGFR
SCHEMBL7987194 0.92 HTR6 (0.37) HTR6CHEK1PDE4BPDE4DEGFR
SCHEMBL7990463 0.92 CHEK1 (0.39) CYP2C19CHEK1EEDACP1
SCHEMBL7990169 0.89 PDE4B (0.37) HTR6PDE4BPDE4DCYP11B1CYP11B2
SCHEMBL7990984 0.88 CCNT1 (0.36) HTR6CYP2C19CHEK1EEDEGFR
SCHEMBL7987981 0.88 EGFR (0.38) CYP2C19CHEK1EEDEGFRABL1
SCHEMBL7976003 0.87 PRKCZ (0.40) HTR6CHEK1PDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed