SCHEMBL7990463

SCHEMBL7990463

COc1cccc(-c2cncc(-c3cn(C(C)C4CCCNC4)c4ccc(C#N)cc34)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 3/20 0.39
KDM1A O60341 2/20 0.36
CYP2C19 P33261 1/20 0.35
FNTA P49354 4/20 0.34
FNTB P49356 4/20 0.34
PGGT1B P53609 3/20 0.34
ACP1 P24666 1/20 0.34
SCN9A Q15858 1/20 0.34
PLAU P00749 1/20 0.34
EED O75530 1/20 0.33
LRRK2 Q5S007 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7975970 0.92 HTR6 (0.39) CHEK1CYP2C19ACP1EED
SCHEMBL7990500 0.91 KDM1A (0.41) CHEK1KDM1ASCN9A
SCHEMBL7505916 0.89 CCNT1 (0.38) KDM1A
SCHEMBL7994923 0.89 PRKCA (0.40) CHEK1CYP2C19ACP1EED
SCHEMBL7975983 0.89 CCNT1 (0.36) KDM1AFNTAFNTB
SCHEMBL7976272 0.89 CCNT1 (0.41) CHEK1CYP2C19ACP1EED
SCHEMBL7990448 0.86 CYP11B1 (0.40) ACP1
SCHEMBL7993914 0.86 HTR6 (0.38) EED
SCHEMBL7994416 0.85 CCNT1 (0.37) KDM1A
SCHEMBL7987194 0.84 HTR6 (0.37) CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed