SCHEMBL8004575

SCHEMBL8004575

N=C(N)NC(=O)OCc1ccc(Oc2cccnc2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.45
SCD O00767 1/20 0.41
SUCNR1 Q9BXA5 1/20 0.40
PPARD Q03181 1/20 0.38
HDAC1 Q13547 3/20 0.37
IDH2 P48735 1/20 0.36
CYP1A2 P05177 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8097516 0.99 SMN1; SMN2 (0.45) SMN1; SMN2SCDSUCNR1PPARDHDAC1
SCHEMBL8004583 0.83 AOC3 (0.49) SMN1; SMN2SUCNR1
Hydrochloric Acid SCHEMBL8104657 0.82 AOC3 (0.50) SMN1; SMN2SUCNR1
SCHEMBL8831863 0.81 SMN1; SMN2 (0.49) SMN1; SMN2
Hydrochloric Acid SCHEMBL8379790 0.80 SMN1; SMN2 (0.48) SMN1; SMN2CYP1A2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL7995076 0.78 PTGDR2 (0.40)
SCHEMBL7995147 0.77 SMN1; SMN2 (0.46) SMN1; SMN2SUCNR1PPARDIDH2CYP1A2
SCHEMBL8185434 0.72 SLC9A1 (0.52) SMN1; SMN2HTR2A
SCHEMBL7995072 0.71 ALDH1A1 (0.53) SMN1; SMN2CYP1A2HTR2AHTR2CHTR2B
Guanidine SCHEMBL8518148 0.70 SMN1; SMN2 (0.46) SMN1; SMN2SUCNR1CYP1A2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748795-B1 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AG (DE) 2000-08-23 EP disclosed
US-6022899-A EFFECTIVE INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-08 US disclosed
US-5753710-A INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-19 US disclosed
EP-0748795-A2 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-18 EP disclosed