SCHEMBL7996580

SCHEMBL7996580

CC1(C)C(=O)N(CCCCN2CCN(c3ccc4ccccc4n3)CC2)CS1(=O)=O

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.63
HTR3A P46098 10/20 0.52
HRH3 Q9Y5N1 2/20 0.52
HTR3E A5X5Y0 1/20 0.52
KDM4E B2RXH2 1/20 0.52
HTR3B O95264 1/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
THPO P40225 1/20 0.52
HTR3D Q70Z44 1/20 0.52
HTR3C Q8WXA8 1/20 0.52
HRH4 Q9H3N8 1/20 0.52
DRD2 P14416 2/20 0.48
DRD3 P35462 1/20 0.48
HTR7 P34969 1/20 0.48
HRH1 P35367 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7996707 0.81 HTR1A (0.63) HTR1AHTR3AHRH3DRD2DRD3
SCHEMBL7993109 0.81 HTR1A (0.61) HTR1AHTR3AHRH3HTR3EKDM4E
SCHEMBL7991688 0.80 RAB9A (0.54) HTR1AHTR3ACYP1A2
SCHEMBL7993335 0.75 HTR1A (0.62) HTR1AHTR3AHRH3DRD2DRD3
SCHEMBL9602546 0.75 HTR1A (0.67) HTR1AHTR3AHRH3HTR3EKDM4E
SCHEMBL7990516 0.74 HTR1A (0.60) HTR1AKDM4EALDH1A1CYP1A2DRD2
SCHEMBL7686047 0.74 HTR1A (0.57) HTR1AHTR3AHRH3HTR3EKDM4E
SCHEMBL7996576 0.73 HTR1A (0.59) HTR1ADRD2HTR7
SCHEMBL3679755 0.73 HTR1A (0.65) HTR1AHTR3AHRH3HTR3EKDM4E
SCHEMBL647772 0.73 HTR1A (0.65) HTR1AHTR3AHRH3HTR3EKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed