SCHEMBL7997544

SCHEMBL7997544

Nc1cc(-c2ccccc2)ccc1C(=O)B1C=CC=C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.50
PPM1B O75688 1/20 0.47
KDM4E B2RXH2 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 1/20 0.47
USP2 O75604 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
HSP90AA1 P07900 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47
HTT P42858 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ACMSD Q8TDX5 3/20 0.45
HNF4A P41235 2/20 0.45
HDAC1 Q13547 3/20 0.42
HDAC3 O15379 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8001505 0.81 AKR1C2 (0.45) IKBKBKDM4ELMNAHSD17B10ACMSD
SCHEMBL2575452 0.79 PPM1B (0.71) IKBKBPPM1BKDM4EKMT2AMAPT
SCHEMBL30456877 0.79 PPM1B (0.71) IKBKBPPM1BKDM4EKMT2AMAPT
SCHEMBL3793566 0.78 IKBKB (0.73) IKBKBPPM1BKDM4EKMT2AMAPT
SCHEMBL3789666 0.76 IKBKB (0.56) IKBKBPPM1BKDM4EKMT2AMAPT
SCHEMBL14392234 0.76 IKBKB (0.56) IKBKBPPM1BKDM4EKMT2AMAPT
SCHEMBL7997824 0.74 DCLRE1B (0.44) IKBKBALDH1A1LMNAACMSDHNF4A
SCHEMBL7994067 0.74 ACLY (0.41) KDM4EKMT2AMAPTMEN1ALDH1A1
SCHEMBL23499274 0.73 PPM1B (0.79) IKBKBPPM1BKDM4EKMT2AMAPT
SCHEMBL29908977 0.73 PPM1B (0.79) IKBKBPPM1BKDM4EKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810858-A4 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN DU PONT PHARM CO (US) 2000-11-15 EP disclosed
EP-0810858-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-12-10 EP disclosed
WO-1996020689-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-11 WO disclosed