SCHEMBL7998527

SCHEMBL7998527

Cc1nnc(CC(C)(C)C/C=C/c2cccc(-c3nn(C)nc3-c3ccccc3)c2)o1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 7/20 0.35
GRIN2B Q13224 7/20 0.35
HDAC1 Q13547 2/20 0.31
HDAC8 Q9BY41 2/20 0.31
HDAC6 Q9UBN7 2/20 0.31
GRN P28799 1/20 0.30
SORT1 Q99523 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8007763 0.86 GRIN1 (0.35) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL7999089 0.84 HDAC1 (0.34) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL7998525 0.82 HDAC1 (0.33) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL8007717 0.81 HDAC6 (0.33) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL10292811 0.79 AAK1 (0.30)
SCHEMBL8007633 0.79 LIPC (0.31) HDAC1HDAC8HDAC6
SCHEMBL10260921 0.79 AAK1 (0.30)
SCHEMBL7998518 0.78 PKM (0.33) HDAC1HDAC8HDAC6
SCHEMBL8013957 0.78 GRIN1 (0.36) GRIN1GRIN2BGRNSORT1
SCHEMBL8010267 0.73 HDAC1 (0.33) HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed