SCHEMBL7999820

SCHEMBL7999820

CC(C)[C@](O)(CCc1ccc(NC(=O)OC(C)(C)C)cc1)CC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.47
DRD2 P14416 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.45
GLS O94925 2/20 0.44
ADAMTS4 O75173 1/20 0.44
PPARG P37231 2/20 0.43
PPARA Q07869 1/20 0.43
MAPK14 Q16539 1/20 0.43
NAMPT P43490 1/20 0.41
SLC13A5 Q86YT5 2/20 0.40
PTPN11 Q06124 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7639674 0.85 ALDH1A1 (0.43) SLC13A5CA1CA2
SCHEMBL7635490 0.85 ALDH1A1 (0.43) SLC13A5CA1CA2
SCHEMBL8008690 0.83 PPARG (0.43) CYP17A1DRD2PTGDR2GLSADAMTS4
SCHEMBL7390375 0.80 CYP17A1 (0.57) CYP17A1DRD2PTGDR2GLSPPARG
SCHEMBL12528285 0.79 CYP17A1 (0.53) CYP17A1DRD2PTGDR2GLSPPARG
SCHEMBL1000732 0.79 NR1H4 (0.58) CYP17A1DRD2PTGDR2GLSPPARG
SCHEMBL20784539 0.78 CYP17A1 (0.54) CYP17A1DRD2PTGDR2GLSADAMTS4
SCHEMBL7998719 0.77 SLC13A5 (0.46) SLC13A5CA2
SCHEMBL7998721 0.77 SLC13A5 (0.46) SLC13A5CA2
SCHEMBL7042995 0.77 DRD2 (0.59) CYP17A1DRD2PTGDR2GLSPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046355-A TOLUENE-4-THIOSULFONIC ACID S-ESTERS AS CHEMICAL INTERMEDIATES FOR VIRICIDES AND ASPARTYL PROTEASE INHIBITORS; AIDS WARNER-LAMBERT COMPANY (US) 2000-04-04 US disclosed
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP disclosed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed