SCHEMBL8008690

SCHEMBL8008690

CCOC(=O)CC(=O)CC(O)(CCc1ccc(NC(=O)OC(C)(C)C)cc1)C(C)C

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.43
PPARA Q07869 1/20 0.43
CYP17A1 P05093 1/20 0.42
DRD2 P14416 1/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
MAPK14 Q16539 1/20 0.38
GLS O94925 1/20 0.38
ADAMTS4 O75173 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
GAA P10253 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PTPRB P23467 1/20 0.38
PPID Q08752 1/20 0.37
NAMPT P43490 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7636689 0.88 PPID (0.49) LMNAMAPTSMN1; SMN2ALDH1A1GAA
SCHEMBL7636702 0.88 PPID (0.49) LMNAMAPTSMN1; SMN2ALDH1A1GAA
SCHEMBL7999820 0.83 CYP17A1 (0.47) PPARGPPARACYP17A1DRD2PTGDR2
SCHEMBL6297746 0.82 CYP4F2 (0.38) PPARGLMNAMAPTALDH1A1HPGD
SCHEMBL6296415 0.82 SMN1; SMN2 (0.44) LMNAMAPTSMN1; SMN2ALDH1A1PPID
SCHEMBL6297611 0.81 PPARG (0.40) PPARGALDH1A1
SCHEMBL3173008 0.80 PPARG (0.53) PPARGPPARACYP17A1DRD2LMNA
SCHEMBL7972075 0.78 CYP4F2 (0.56) PPARGPPARACYP17A1DRD2LMNA
SCHEMBL6303036 0.78 ALDH1A1 (0.37) ALDH1A1HPGD
SCHEMBL8345213 0.76 LMNA (0.50) PPARGPPARALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046355-A TOLUENE-4-THIOSULFONIC ACID S-ESTERS AS CHEMICAL INTERMEDIATES FOR VIRICIDES AND ASPARTYL PROTEASE INHIBITORS; AIDS WARNER-LAMBERT COMPANY (US) 2000-04-04 US disclosed
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP disclosed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed