SCHEMBL8007166

SCHEMBL8007166

Cc1cc(-c2ccc(Cl)cn2)ccc1CO

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.44
BACE1 P56817 2/20 0.38
GRIA2 P42262 1/20 0.38
S1PR1 P21453 1/20 0.38
CNR2 P34972 1/20 0.38
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PDXK O00764 1/20 0.36
NOTUM Q6P988 2/20 0.36
HSD17B1 P14061 2/20 0.35
HSD17B2 P37059 2/20 0.35
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16385303 0.80 HSD17B1 (0.52) P2RX7BACE1GRIA2S1PR1CNR2
SCHEMBL8023947 0.79 PTGER4 (0.48) P2RX7S1PR1
SCHEMBL14524935 0.79 ALOX5 (0.44) S1PR1GRIN1GRIN2BNOTUM
SCHEMBL7941960 0.78 P2RX7 (0.46) P2RX7S1PR1GRIN1GRIN2BHDAC1
SCHEMBL8028548 0.78 KDM4E (0.47) P2RX7GRIN1GRIN2BKDM1A
SCHEMBL25480188 0.75 CYP2D6 (0.45) S1PR1
SCHEMBL21753409 0.75 CBFB (0.44) P2RX7S1PR1
SCHEMBL1096478 0.74 PSEN1 (0.42) P2RX7HDAC3HDAC1HDAC2HDAC6
SCHEMBL16385279 0.74 KDM4E (0.48) KDM1A
SCHEMBL12970151 0.74 KDM1A (0.53) CNR2NOTUMKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071504-A1 2,6-DISUBSTITUTED PYRIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed