SCHEMBL8028548

SCHEMBL8028548

Cc1cc(-c2ccc(C#N)cn2)ccc1CO

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
HPGD P15428 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
HTT P42858 1/20 0.47
AR P10275 4/20 0.43
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
P2RX7 Q99572 1/20 0.40
GRM5 P41594 3/20 0.39
KDM1A O60341 1/20 0.37
EGLN2 Q96KS0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3997043 0.81 MMP3 (0.46) ALDH1A1ARGRIN1GRIN2B
SCHEMBL8007166 0.78 P2RX7 (0.44) GRIN1GRIN2BP2RX7KDM1A
SCHEMBL410177 0.77 CYP2A6 (0.41) ALDH1A1AR
SCHEMBL8019866 0.76 KDM4E (0.54) KDM4EALDH1A1HPGDL3MBTL1HTT
SCHEMBL29818872 0.76 KDM4E (0.54) KDM4EALDH1A1HPGDL3MBTL1HTT
SCHEMBL8023947 0.76 PTGER4 (0.48) KDM4EALDH1A1P2RX7
SCHEMBL8028511 0.75 HRH2 (0.42) AREGLN2
SCHEMBL3467724 0.75 CYP11B1 (0.47) KDM4EALDH1A1HPGDL3MBTL1HTT
SCHEMBL3718441 0.75 KDM4E (0.47) KDM4EALDH1A1HPGDL3MBTL1HTT
SCHEMBL7941960 0.75 P2RX7 (0.46) KDM4EL3MBTL1GRIN1GRIN2BP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071504-A1 2,6-DISUBSTITUTED PYRIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed