SCHEMBL8009329

SCHEMBL8009329

CCc1ccccc1NC=C1C(=O)N(c2ccc(S(=O)(=O)N(CC)CC)cc2)N=C1C(CC)C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SHMT2 P34897 1/20 0.37
ALDH1A1 P00352 4/20 0.36
TP53 P04637 2/20 0.36
MAPT P10636 1/20 0.36
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
HTT P42858 1/20 0.35
RECQL P46063 1/20 0.35
PKM P14618 1/20 0.34
KMT2A Q03164 1/20 0.34
PHOSPHO1 Q8TCT1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008689 0.89 THRB (0.40) SHMT2ALDH1A1MAPTNPC1HPGD
SCHEMBL8009344 0.85 MAPT (0.43) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL8008606 0.85 KDM4E (0.35) ALDH1A1MAPTHPGDHTTKMT2A
SCHEMBL6952092 0.84 MAPT (0.39) SHMT2ALDH1A1TP53MAPTNPC1
SCHEMBL6952098 0.84 MAPT (0.39) SHMT2ALDH1A1TP53MAPTNPC1
SCHEMBL8011512 0.84 MEN1 (0.39) ALDH1A1MAPTNPC1HPGDRAB9A
SCHEMBL6947265 0.83 KAT8 (0.42) ALDH1A1MAPTHPGDSMN1; SMN2HTT
SCHEMBL6947262 0.83 KAT8 (0.42) ALDH1A1MAPTHPGDSMN1; SMN2HTT
SCHEMBL8008615 0.82 KMT2A (0.35) ALDH1A1MAPTNPC1HPGDRAB9A
SCHEMBL8009323 0.81 MAPT (0.37) SHMT2ALDH1A1TP53MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6034099-A Method for inhibiting neoplastic lesions by administering 4-(arylmethylene)- 2, 3- dihydro-pyrazol-3-ones CELL PATHWAYS, INC. (US) 2000-03-07 US claimed
US-6034099-A Method for inhibiting neoplastic lesions by administering 4-(arylmethylene)- 2, 3- dihydro-pyrazol-3-ones CELL PATHWAYS, INC. (US) 2000-03-07 US disclosed