SCHEMBL8017476

SCHEMBL8017476

COc1ccccc1C1CNCCN1CCNc1ccncc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.41
HTR2A P28223 1/20 0.41
HTR2B P41595 1/20 0.41
HTR1A P08908 2/20 0.36
ADRA1A P35348 1/20 0.36
GSK3B P49841 4/20 0.36
DRD2 P14416 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
AKT1 P31749 1/20 0.34
CHRNA7 P36544 1/20 0.34
TSHR P16473 1/20 0.34
ALOX12 P18054 1/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
ADRB1 P08588 1/20 0.34
CYP2C19 P33261 1/20 0.34
DRD3 P35462 1/20 0.34
HTR3A P46098 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5915126 0.80 DRD2 (0.51) HTR2CHTR2AHTR2BHTR1ADRD2
SCHEMBL9527372 0.76 HTR2C (0.46) HTR2CHTR2AHTR2BDRD2SLC6A2
SCHEMBL1074633 0.73 HTR2C (0.47) HTR2CHTR2AHTR2BHTR1ADRD2
SCHEMBL4125113 0.73 HTR2C (0.39) HTR2CHTR2AHTR2BHTR1AADRA1A
SCHEMBL8055769 0.72 HRH1 (0.56) HTR2CHTR2AHTR2BHTR1AADRA1A
SCHEMBL27526873 0.72 CYP3A4 (0.39) GSK3BCHRNA7SIGMAR1
SCHEMBL8422421 0.70 HTR2C (0.43) HTR2CHTR2AHTR2BSLC6A2SLC6A4
SCHEMBL8911446 0.69 HTR2C (0.53) HTR2CHTR2AHTR2BDRD2HTR3E
SCHEMBL2429178 0.68 HTR1A (0.51) HTR1AADRA1ATSHRCYP2C19
SCHEMBL8422451 0.67 HTR2B (0.44) HTR2CHTR2AHTR2BHTR1ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127357-A N-((phenyl, benzodioxinyl or N-heteroarylpiperazinyl)alkyl)-N-(N-heteroaryl)substituted carboxamides JOHN WYETH & BROTHER, LTD. (GB) 2000-10-03 US disclosed