SCHEMBL8019456

SCHEMBL8019456

CNc1nc2c(S(=O)(=O)c3ccc(F)cc3)nnn2c2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.64
HPGD P15428 7/20 0.64
ALDH1A1 P00352 8/20 0.63
GAA P10253 4/20 0.63
KMT2A Q03164 2/20 0.63
RXFP1 Q9HBX9 5/20 0.62
NPSR1 Q6W5P4 2/20 0.62
MAPT P10636 7/20 0.61
RECQL P46063 1/20 0.61
POLB P06746 2/20 0.60
HTR6 P50406 4/20 0.58
PKM P14618 1/20 0.55
CRHBP P24387 1/20 0.53
CRHR2 Q13324 1/20 0.53
TP53 P04637 1/20 0.53
MEN1 O00255 1/20 0.51
THRB P10828 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8021786 0.91 KDM4E (0.72) KDM4EHPGDALDH1A1GAAKMT2A
SCHEMBL8021789 0.88 KDM4E (0.64) KDM4EHPGDALDH1A1GAAKMT2A
SCHEMBL8019479 0.86 HPGD (0.60) KDM4EHPGDALDH1A1GAAKMT2A
SCHEMBL8018281 0.82 HPGD (0.53) KDM4EHPGDALDH1A1GAAKMT2A
SCHEMBL8026556 0.82 KDM4E (0.64) KDM4EHPGDALDH1A1GAAKMT2A
SCHEMBL8031028 0.81 MAPT (0.71) KDM4EALDH1A1GAAKMT2ARXFP1
SCHEMBL8021777 0.81 HTR6 (0.56) RXFP1MAPTPOLBHTR6TP53
SCHEMBL8018835 0.79 HPGD (0.69) KDM4EHPGDALDH1A1GAAKMT2A
SCHEMBL8031022 0.79 HTR6 (0.72) KDM4EHPGDALDH1A1GAAKMT2A
SCHEMBL8031518 0.78 RXFP1 (0.70) KDM4EHPGDALDH1A1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed