SCHEMBL8021789

SCHEMBL8021789

CNc1nc2c(S(=O)(=O)c3cccc(F)c3)nnn2c2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.64
HPGD P15428 5/20 0.64
MAPT P10636 8/20 0.63
ALDH1A1 P00352 6/20 0.63
RECQL P46063 1/20 0.63
RXFP1 Q9HBX9 4/20 0.62
NPSR1 Q6W5P4 2/20 0.62
GAA P10253 4/20 0.60
KMT2A Q03164 2/20 0.60
POLB P06746 1/20 0.57
TP53 P04637 2/20 0.55
HTR6 P50406 3/20 0.53
THRB P10828 2/20 0.51
PKM P14618 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8019456 0.88 KDM4E (0.64) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8021786 0.88 KDM4E (0.72) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8026556 0.88 KDM4E (0.64) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8019463 0.83 HPGD (0.53) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8028518 0.83 HTR6 (0.55) MAPTRXFP1GAATP53HTR6
SCHEMBL8027148 0.78 RXFP1 (0.65) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8019479 0.77 HPGD (0.60) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8021669 0.77 HPGD (0.45) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8030786 0.77 RXFP1 (0.65) KDM4EHPGDMAPTALDH1A1RECQL
SCHEMBL8031022 0.76 HTR6 (0.72) KDM4EHPGDMAPTALDH1A1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed