SCHEMBL8019463

SCHEMBL8019463

CN(C)c1nc2c(S(=O)(=O)c3cccc(F)c3)nnn2c2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.53
KDM4E B2RXH2 6/20 0.53
ALDH1A1 P00352 6/20 0.53
MAPT P10636 3/20 0.53
RECQL P46063 1/20 0.53
RXFP1 Q9HBX9 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
GAA P10253 3/20 0.50
KMT2A Q03164 1/20 0.50
TP53 P04637 2/20 0.48
POLB P06746 1/20 0.48
HTR6 P50406 5/20 0.47
CRHBP P24387 2/20 0.46
CRHR2 Q13324 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8018281 0.88 HPGD (0.53) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8018278 0.88 HPGD (0.60) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8027148 0.88 RXFP1 (0.65) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8019460 0.88 HTR6 (0.60) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8021789 0.83 KDM4E (0.64) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8018356 0.83 HTR6 (0.48) MAPTRXFP1GAAHTR6
SCHEMBL8034001 0.79 RXFP1 (0.62) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8021669 0.77 HPGD (0.45) HPGDKDM4EALDH1A1MAPTRECQL
SCHEMBL8030787 0.77 RXFP1 (0.57) MAPTRXFP1GAATP53HTR6
SCHEMBL8029045 0.76 KDM4E (0.61) HPGDKDM4EALDH1A1MAPTRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093934-A2 SUBSTITUTED 3-SULPHONYL-[1,2,3]TRIAZOLO [1,5-A]PYRIMIDINES-ANTAGONISTS OF SEROTONIN 5-HT6 RECEPTORS, MEDICINAL SUBSTANCE, PHARMACEUTICAL COMPOSITION, MEDICINAL PREPARATION AND METHODS FOR THE PRODUCTION THEREOF ALLA CHEM, LLC (US) 2009-07-30 WO disclosed